Reaction Details |
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Target | Cannabinoid receptor 2 |
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Ligand | BDBM76051 |
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Substrate/Competitor | n/a |
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Meas. Tech. | SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 |
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IC50 | >32000±n/a nM |
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Citation | PubChem, PC SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Cannabinoid receptor 2 |
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Name: | Cannabinoid receptor 2 |
Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 39690.94 |
Organism: | Homo sapiens (Human) |
Description: | P34972 |
Residue: | 360 |
Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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BDBM76051 |
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n/a |
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Name | BDBM76051 |
Synonyms: | 2-azanylidene-N,1-dicyclopentyl-8-methyl-5-oxidanylidene-dipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | MLS-0437148.0001 | N,1-dicyclopentyl-2-imino-5-keto-8-methyl-dipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | N,1-dicyclopentyl-2-imino-8-methyl-5-oxo-3-dipyrido[1,2-d:3',4'-f]pyrimidinecarboxamide | N,1-dicyclopentyl-2-imino-8-methyl-5-oxodipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | cid_3151387 |
Type | Small organic molecule |
Emp. Form. | C23H27N5O2 |
Mol. Mass. | 405.4928 |
SMILES | Cc1ccc2nc3n(C4CCCC4)c(=N)c(cc3c(=O)n2c1)C(=O)NC1CCCC1 |
Structure |
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