| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
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| Ligand | BDBM76033 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 |
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| EC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 35 |
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| Name: | G-protein coupled receptor 35 |
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| Synonyms: | G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 34085.57 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_33695097 |
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| Residue: | 309 |
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| Sequence: | MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
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| BDBM76033 |
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| n/a |
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| Name | BDBM76033 |
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| Synonyms: | 4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-N-(phenylmethyl)-1-piperazinecarboxamide | 4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-N-(phenylmethyl)piperazine-1-carboxamide | MLS-0437132.0001 | N-benzyl-4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)piperazine-1-carboxamide | N-benzyl-4-(2-methyl-5,6,7,8-tetrahydrobenzothiopheno[2,3-d]pyrimidin-4-yl)piperazine-1-carboxamide | cid_1468079 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H27N5OS |
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| Mol. Mass. | 421.558 |
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| SMILES | Cc1nc(N2CCN(CC2)C(=O)NCc2ccccc2)c2c3CCCCc3sc2n1 |
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| Structure | 
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