| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 55 |
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| Ligand | BDBM76048 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 4 |
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| IC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 4 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 55 |
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| Name: | G-protein coupled receptor 55 |
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| Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36649.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1292265 |
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| Residue: | 319 |
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| Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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| BDBM76048 |
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| n/a |
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| Name | BDBM76048 |
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| Synonyms: | 1-cyclopentyl-2-imino-5-keto-N-(2-morpholinoethyl)dipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | 1-cyclopentyl-2-imino-N-(2-morpholin-4-ylethyl)-5-oxodipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | 1-cyclopentyl-2-imino-N-[2-(4-morpholinyl)ethyl]-5-oxo-3-dipyrido[1,2-d:3',4'-f]pyrimidinecarboxamide | 2-azanylidene-1-cyclopentyl-N-(2-morpholin-4-ylethyl)-5-oxidanylidene-dipyrido[1,2-d:3',4'-f]pyrimidine-3-carboxamide | MLS-0437145.0001 | cid_1050206 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H28N6O3 |
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| Mol. Mass. | 436.5068 |
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| SMILES | N=c1c(cc2c(nc3ccccn3c2=O)n1C1CCCC1)C(=O)NCCN1CCOCC1 |
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| Structure | 
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