| Reaction Details |
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 | Report a problem with these data |
| Target | Sentrin-specific protease 8 |
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| Ligand | BDBM76367 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
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| IC50 | 2670±n/a nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Sentrin-specific protease 8 |
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| Name: | Sentrin-specific protease 8 |
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| Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 24104.52 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_262118306 |
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| Residue: | 212 |
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| Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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| BDBM76367 |
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| n/a |
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| Name | BDBM76367 |
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| Synonyms: | MLS000065767 | N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-methyl-3-furamide | N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-methyl-3-furancarboxamide | N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-methyl-furan-3-carboxamide | N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-methylfuran-3-carboxamide | SMR000080448 | cid_1245882 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H17N3O2S |
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| Mol. Mass. | 291.369 |
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| SMILES | Cc1occc1C(=O)Nc1nnc(s1)C1CCCCC1 |
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| Structure | 
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