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TargetSentrin-specific protease 8
LigandBDBM76369
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50 1560±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sentrin-specific protease 8
Name:Sentrin-specific protease 8
Synonyms:DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:Enzyme Catalytic Domain
Mol. Mass.:24104.52
Organism:Homo sapiens (Human)
Description:gi_262118306
Residue:212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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  Blast E-value cutoff:
BDBM76369
n/a
NameBDBM76369
Synonyms:MLS000100578 | N-(1,3-benzothiazol-2-yl)-5-chloranyl-thiophene-2-carboxamide | N-(1,3-benzothiazol-2-yl)-5-chloro-2-thiophenecarboxamide | N-(1,3-benzothiazol-2-yl)-5-chloro-thiophene-2-carboxamide | N-(1,3-benzothiazol-2-yl)-5-chlorothiophene-2-carboxamide | SMR000017422 | cid_2414873
TypeSmall organic molecule
Emp. Form.C12H7ClN2OS2
Mol. Mass.294.78
SMILESClc1ccc(s1)C(=O)Nc1nc2ccccc2s1
Structure
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