Reaction Details |
| Report a problem with these data |
Target | Sentrin-specific protease 8 |
---|
Ligand | BDBM76524 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
---|
IC50 | 1880±n/a nM |
---|
Citation | PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
Sentrin-specific protease 8 |
---|
Name: | Sentrin-specific protease 8 |
Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 24104.52 |
Organism: | Homo sapiens (Human) |
Description: | gi_262118306 |
Residue: | 212 |
Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
|
|
|
BDBM76524 |
---|
n/a |
---|
Name | BDBM76524 |
Synonyms: | 4-[(4-methyl-5-phenyl-1,3-thiazol-2-yl)amino]benzoic acid | 4-[(4-methyl-5-phenyl-2-thiazolyl)amino]benzoic acid | 4-[(4-methyl-5-phenyl-thiazol-2-yl)amino]benzoic acid | MLS000408851 | SMR000243082 | cid_2384167 |
Type | Small organic molecule |
Emp. Form. | C17H14N2O2S |
Mol. Mass. | 310.37 |
SMILES | Cc1nc(Nc2ccc(cc2)C(O)=O)sc1-c1ccccc1 |
Structure |
|