| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Sentrin-specific protease 8 |
|---|
| Ligand | BDBM76569 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
|---|
| IC50 | 1830±n/a nM |
|---|
| Citation |  PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Sentrin-specific protease 8 |
|---|
| Name: | Sentrin-specific protease 8 |
|---|
| Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 24104.52 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_262118306 |
|---|
| Residue: | 212 |
|---|
| Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
|
|
|
|---|
| BDBM76569 |
|---|
| n/a |
|---|
| Name | BDBM76569 |
|---|
| Synonyms: | (3Z)-1-ethyl-3-(2-quinolinylhydrazinylidene)-2-indolone | (3Z)-1-ethyl-3-(2-quinolylhydrazono)oxindole | (3Z)-1-ethyl-3-(quinolin-2-ylhydrazinylidene)indol-2-one | 1-Ethyl-3-(quinolin-2-yl-hydrazono)-1,3-dihydro-indol-2-one | MLS000778542 | SMR000415336 | cid_6040562 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H16N4O |
|---|
| Mol. Mass. | 316.3565 |
|---|
| SMILES | CCN1C(=O)C(=NNc2ccc3ccccc3n2)c2ccccc12 |w:6.6| |
|---|
| Structure | 
|
|---|
Search and Browse
