| Reaction Details |
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 | Report a problem with these data |
| Target | Sentrin-specific protease 8 |
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| Ligand | BDBM76674 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
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| IC50 | 2580±n/a nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Sentrin-specific protease 8 |
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| Name: | Sentrin-specific protease 8 |
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| Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 24104.52 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_262118306 |
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| Residue: | 212 |
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| Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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| BDBM76674 |
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| n/a |
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| Name | BDBM76674 |
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| Synonyms: | 4-(4-Chloro-phenylazo)-3-methyl-5-oxo-4,5-dihydro-pyrazole-1-carbothioic acid amide | 4-(4-chlorophenyl)azo-3-methyl-5-oxo-4H-pyrazole-1-carbothioamide | 4-(4-chlorophenyl)azo-5-keto-3-methyl-2-pyrazoline-1-carbothioamide | 4-[(4-chlorophenyl)diazenyl]-3-methyl-5-oxidanylidene-4H-pyrazole-1-carbothioamide | 4-[(4-chlorophenyl)diazenyl]-3-methyl-5-oxo-4H-pyrazole-1-carbothioamide | MLS001202823 | SMR000513810 | cid_3103951 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H10ClN5OS |
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| Mol. Mass. | 295.748 |
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| SMILES | Cc1[nH]n(C(N)=S)c(=O)c1N=Nc1ccc(Cl)cc1 |w:10.10| |
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| Structure | 
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