| Reaction Details |
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 | Report a problem with these data |
| Target | X-box-binding protein 1 |
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| Ligand | BDBM67807 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | XBP1 DR counterscreen for CHOP |
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| IC50 | 290±n/a nM |
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| Citation |  PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| X-box-binding protein 1 |
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| Name: | X-box-binding protein 1 |
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| Synonyms: | TREB5 | XBP1 | XBP1_HUMAN | XBP2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 28704.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_47678753 |
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| Residue: | 261 |
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| Sequence: | MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARK
RQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLR
EKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQL
SPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVP
YQPPFLCQWGRHQPSWKPLMN
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| BDBM67807 |
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| n/a |
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| Name | BDBM67807 |
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| Synonyms: | 5-(4-methylbenzyl)-7-(trifluoromethyl)-3,3a-dihydro-1H-thiazolo[3,4-a]quinoxalin-4-one | 5-(4-methylbenzyl)-7-(trifluoromethyl)-3,3a-dihydro[1,3]thiazolo[3,4-a]quinoxalin-4(5H)-one | 5-[(4-methylphenyl)methyl]-7-(trifluoromethyl)-3,3a-dihydro-1H-[1,3]thiazolo[3,4-a]quinoxalin-4-one | 5-[(4-methylphenyl)methyl]-7-(trifluoromethyl)-3,3a-dihydro-1H-thiazolo[3,4-a]quinoxalin-4-one | MLS000541396 | SMR000126254 | cid_3806160 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H17F3N2OS |
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| Mol. Mass. | 378.411 |
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| SMILES | Cc1ccc(CN2C(=O)C3CSCN3c3ccc(cc23)C(F)(F)F)cc1 |
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| Structure | 
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