| Reaction Details |
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 | Report a problem with these data |
| Target | X-box-binding protein 1 |
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| Ligand | BDBM61434 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | XBP1 DR counterscreen for CHOP |
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| IC50 | 160±n/a nM |
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| Citation |  PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| X-box-binding protein 1 |
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| Name: | X-box-binding protein 1 |
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| Synonyms: | TREB5 | XBP1 | XBP1_HUMAN | XBP2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 28704.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_47678753 |
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| Residue: | 261 |
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| Sequence: | MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARK
RQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLR
EKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQL
SPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVP
YQPPFLCQWGRHQPSWKPLMN
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| BDBM61434 |
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| n/a |
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| Name | BDBM61434 |
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| Synonyms: | 3'-(4-fluorophenyl)-4,4,6,8-tetramethyl-4H,4'H-spiro[pyrrolo[3,2,1-ij]quinoline-1,2'-[1,3]thiazolidine]-2,4'-dione | MLS000538872 | SMR000144709 | cid_2981819 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H21FN2O2S |
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| Mol. Mass. | 408.488 |
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| SMILES | CC1=CC(C)(C)N2C(=O)C3(SCC(=O)N3c3ccc(F)cc3)c3cc(C)cc1c23 |t:1| |
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| Structure | 
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