| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Perilipin-1 |
|---|
| Ligand | BDBM79412 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain |
|---|
| IC50 | 5597±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-1 (PLIN1) (2K validation set) PubChem Bioassay(2011)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Perilipin-1 |
|---|
| Name: | Perilipin-1 |
|---|
| Synonyms: | PERI | PLIN | PLIN1 | PLIN1_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 55988.69 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_223718203 |
|---|
| Residue: | 522 |
|---|
| Sequence: | MAVNKGLTLLDGDLPEQENVLQRVLQLPVVSGTCECFQKTYTSTKEAHPLVASVCNAYEK
GVQSASSLAAWSMEPVVRRLSTQFTAANELACRGLDHLEEKIPALQYPPEKIASELKDTI
STRLRSARNSISVPIASTSDKVLGAALAGCELAWGVARDTAEFAANTRAGRLASGGADLA
LGSIEKVVEYLLPPDKEESAPAPGHQQAQKSPKAKPSLLSRVGALTNTLSRYTVQTMARA
LEQGHTVAMWIPGVVPLSSLAQWGASVAMQAVSRRRSEVRVPWLHSLAAAQEEDHEDQTD
TEGEDTEEEEELETEENKFSEVAALPGPRGLLGGVAHTLQKTLQTTISAVTWAPAAVLGM
AGRVLHLTPAPAVSSTKGRAMSLSDALKGVTDNVVDTVVHYVPLPRLSLMEPESEFRDID
NPPAEVERREAERRASGAPSAGPEPAPRLAQPRRSLRSAQSPGAPPGPGLEDEVATPAAP
RPGFPAVPREKPKRRVSDSFFRPSVMEPILGRTHYSQLRKKS
|
|
|
|---|
| BDBM79412 |
|---|
| n/a |
|---|
| Name | BDBM79412 |
|---|
| Synonyms: | (2E,5E)-2,5-bis(3,4-dimethoxybenzylidene)cyclopentanone | (2E,5E)-2,5-bis[(3,4-dimethoxyphenyl)methylidene]-1-cyclopentanone | (2E,5E)-2,5-bis[(3,4-dimethoxyphenyl)methylidene]cyclopentan-1-one | (2E,5E)-2,5-diveratrylidenecyclopentanone | MLS000586404 | SMR000204767 | cid_5714141 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H24O5 |
|---|
| Mol. Mass. | 380.4337 |
|---|
| SMILES | COc1ccc(\C=C2/CC\C(=C/c3ccc(OC)c(OC)c3)C2=O)cc1OC |
|---|
| Structure | 
|
|---|
Search and Browse
