| Reaction Details |
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 | Report a problem with these data |
| Target | Perilipin-1 |
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| Ligand | BDBM79425 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain |
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| IC50 | 4420±n/a nM |
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| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-1 (PLIN1) (2K validation set) PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Perilipin-1 |
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| Name: | Perilipin-1 |
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| Synonyms: | PERI | PLIN | PLIN1 | PLIN1_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 55988.69 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_223718203 |
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| Residue: | 522 |
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| Sequence: | MAVNKGLTLLDGDLPEQENVLQRVLQLPVVSGTCECFQKTYTSTKEAHPLVASVCNAYEK
GVQSASSLAAWSMEPVVRRLSTQFTAANELACRGLDHLEEKIPALQYPPEKIASELKDTI
STRLRSARNSISVPIASTSDKVLGAALAGCELAWGVARDTAEFAANTRAGRLASGGADLA
LGSIEKVVEYLLPPDKEESAPAPGHQQAQKSPKAKPSLLSRVGALTNTLSRYTVQTMARA
LEQGHTVAMWIPGVVPLSSLAQWGASVAMQAVSRRRSEVRVPWLHSLAAAQEEDHEDQTD
TEGEDTEEEEELETEENKFSEVAALPGPRGLLGGVAHTLQKTLQTTISAVTWAPAAVLGM
AGRVLHLTPAPAVSSTKGRAMSLSDALKGVTDNVVDTVVHYVPLPRLSLMEPESEFRDID
NPPAEVERREAERRASGAPSAGPEPAPRLAQPRRSLRSAQSPGAPPGPGLEDEVATPAAP
RPGFPAVPREKPKRRVSDSFFRPSVMEPILGRTHYSQLRKKS
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| BDBM79425 |
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| n/a |
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| Name | BDBM79425 |
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| Synonyms: | 8-[(E)-3-(2-hydroxy-4-methoxy-phenyl)-3-keto-prop-1-enyl]-4H-1,3-benzodioxin-6-carboxylic acid | 8-[(E)-3-(2-hydroxy-4-methoxyphenyl)-3-oxoprop-1-enyl]-4H-1,3-benzodioxin-6-carboxylic acid | 8-[(E)-3-(2-hydroxy-4-methoxyphenyl)-3-oxoprop-1-enyl]-4H-1,3-benzodioxine-6-carboxylic acid | 8-[(E)-3-(4-methoxy-2-oxidanyl-phenyl)-3-oxidanylidene-prop-1-enyl]-4H-1,3-benzodioxine-6-carboxylic acid | MLS000774889 | SMR000368141 | cid_5926982 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H16O7 |
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| Mol. Mass. | 356.3261 |
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| SMILES | COc1ccc(C(=O)\C=C\c2cc(cc3COCOc23)C(O)=O)c(O)c1 |
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| Structure | 
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