| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Perilipin-1 |
|---|
| Ligand | BDBM34651 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain |
|---|
| IC50 | >79476±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-1 (PLIN1) (2K validation set) PubChem Bioassay(2011)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Perilipin-1 |
|---|
| Name: | Perilipin-1 |
|---|
| Synonyms: | PERI | PLIN | PLIN1 | PLIN1_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 55988.69 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_223718203 |
|---|
| Residue: | 522 |
|---|
| Sequence: | MAVNKGLTLLDGDLPEQENVLQRVLQLPVVSGTCECFQKTYTSTKEAHPLVASVCNAYEK
GVQSASSLAAWSMEPVVRRLSTQFTAANELACRGLDHLEEKIPALQYPPEKIASELKDTI
STRLRSARNSISVPIASTSDKVLGAALAGCELAWGVARDTAEFAANTRAGRLASGGADLA
LGSIEKVVEYLLPPDKEESAPAPGHQQAQKSPKAKPSLLSRVGALTNTLSRYTVQTMARA
LEQGHTVAMWIPGVVPLSSLAQWGASVAMQAVSRRRSEVRVPWLHSLAAAQEEDHEDQTD
TEGEDTEEEEELETEENKFSEVAALPGPRGLLGGVAHTLQKTLQTTISAVTWAPAAVLGM
AGRVLHLTPAPAVSSTKGRAMSLSDALKGVTDNVVDTVVHYVPLPRLSLMEPESEFRDID
NPPAEVERREAERRASGAPSAGPEPAPRLAQPRRSLRSAQSPGAPPGPGLEDEVATPAAP
RPGFPAVPREKPKRRVSDSFFRPSVMEPILGRTHYSQLRKKS
|
|
|
|---|
| BDBM34651 |
|---|
| n/a |
|---|
| Name | BDBM34651 |
|---|
| Synonyms: | Amrinon | Amrinone | CHEMBL12856 | Cordemcura | INAMRINONE | Inocor | MLS000069829 | SMR000058850 | Win40680 | Wincoram | cid_3698 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C10H9N3O |
|---|
| Mol. Mass. | 187.198 |
|---|
| SMILES | Nc1cc(c[nH]c1=O)-c1ccncc1 |
|---|
| Structure | 
|
|---|
Search and Browse
