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TargetTropomyosin alpha-1 chain
LigandBDBM79651
Substrate/Competitorn/a
Meas. Tech.Fluorescence-based biochemical high throughput dose response assay for activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF)
EC50>71507±n/a nM
Citation PubChem, PC Fluorescence-based biochemical high throughput dose response assay for activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF) PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Tropomyosin alpha-1 chain
Name:Tropomyosin alpha-1 chain
Synonyms:TPM1 | TPM1_PIG | cardiac alpha tropomyosin
Type:Enzyme Catalytic Domain
Mol. Mass.:32681.01
Organism:Sus scrofa
Description:P42639
Residue:284
Sequence:
MDAIKKKMQMLKLDKENALDRAEQAEADKKAAEDRSKRLEDELVSLQKKLKATEDELDKY
SEAPKDAQEKLELAEKKATDAEADVASLNRRIQLVEEELDRAQERLATALQKLEEAEKAA
DESERGMKVIESRAQKDEEKMEIQEIQLKEAKHIAEDADRKYEEVARKLVIIESDLERAE
ERAELSEGKCAELEEELKTVTNNLKSLEAQAEKYSQKEDKYEEEIKVLSDKLKEAETRAE
FAERSVTKLEKSIDDLEDELYAQKLKYKAISEELDHALNDMTSI
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  Blast E-value cutoff:
BDBM79651
n/a
NameBDBM79651
Synonyms:1-(2-furoyl)-4-[3-(phenylthio)propanoyl]piperazine | 1-[4-(2-furoyl)piperazino]-3-(phenylthio)propan-1-one | 1-[4-(furan-2-carbonyl)piperazin-1-yl]-3-phenylsulfanylpropan-1-one | 1-[4-(furan-2-ylcarbonyl)piperazin-1-yl]-3-phenylsulfanyl-propan-1-one | 1-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3-(phenylthio)-1-propanone | MLS000066424 | SMR000081380 | cid_2229128
TypeSmall organic molecule
Emp. Form.C18H20N2O3S
Mol. Mass.344.428
SMILESO=C(CCSc1ccccc1)N1CCN(CC1)C(=O)c1ccco1
Structure
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