Reaction Details |
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Target | Orexin/Hypocretin receptor type 1 |
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Ligand | BDBM79850 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Homogeneous Time Resolved Fluorescence (HTRF)-based cell-based high throughput dose response assay for antagonists of the orexin 1 receptor (OX1R; HCRTR1) |
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IC50 | 1241±n/a nM |
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Citation | PubChem, PC Homogeneous Time Resolved Fluorescence (HTRF)-based cell-based high throughput dose response assay for antagonists of the orexin 1 receptor (OX1R; HCRTR1) PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Orexin/Hypocretin receptor type 1 |
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Name: | Orexin/Hypocretin receptor type 1 |
Synonyms: | HCRTR1 | Hypocretin receptor type 1 | OX1R_HUMAN | Orexin receptor type 1 | Orexin receptor type 1 (OR 1) | Orexin receptor type 1 (OR-1) | Orexin receptor type 1 (OX1) | Orexin receptor type 1 (OX1R) | Orexin receptor type 1 (OxR1) | Ox1r |
Type: | Protein |
Mol. Mass.: | 47554.50 |
Organism: | Homo sapiens (Human) |
Description: | O43613 |
Residue: | 425 |
Sequence: | MEPSATPGAQMGVPPGSREPSPVPPDYEDEFLRYLWRDYLYPKQYEWVLIAAYVAVFVVA
LVGNTLVCLAVWRNHHMRTVTNYFIVNLSLADVLVTAICLPASLLVDITESWLFGHALCK
VIPYLQAVSVSVAVLTLSFIALDRWYAICHPLLFKSTARRARGSILGIWAVSLAIMVPQA
AVMECSSVLPELANRTRLFSVCDERWADDLYPKIYHSCFFIVTYLAPLGLMAMAYFQIFR
KLWGRQIPGTTSALVRNWKRPSDQLGDLEQGLSGEPQPRARAFLAEVKQMRARRKTAKML
MVVLLVFALCYLPISVLNVLKRVFGMFRQASDREAVYACFTFSHWLVYANSAANPIIYNF
LSGKFREQFKAAFSCCLPGLGPCGSLKAPSPRSSASHKSLSLQSRCSISKISEHVVLTSV
TTVLP
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BDBM79850 |
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n/a |
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Name | BDBM79850 |
Synonyms: | (fluoren-9-ylideneamino) 3,4-dimethoxybenzoate | 3,4-dimethoxybenzoic acid (9-fluorenylideneamino) ester | 3,4-dimethoxybenzoic acid (fluoren-9-ylideneamino) ester | 9H-fluoren-9-one O-(3,4-dimethoxybenzoyl)oxime | MLS000576487 | SMR000185871 | cid_1813635 |
Type | Small organic molecule |
Emp. Form. | C22H17NO4 |
Mol. Mass. | 359.3747 |
SMILES | [#6]-[#8]-c1ccc(cc1-[#8]-[#6])-[#6](=O)-[#8]\[#7]=[#6]-1/c2ccccc2-c2ccccc-12 |
Structure |
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