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TargetDNA dC->dU-editing enzyme APOBEC-3A
LigandBDBM59578
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of APOBEC3G DNA Deaminase Inhibitors via a A3A counterscreen
Temperature298.15±n/a K
IC50>100000±n/a nM
Commentsextracted
Citation PubChem, PC Dose Response confirmation of APOBEC3G DNA Deaminase Inhibitors via a A3A counterscreen PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
DNA dC->dU-editing enzyme APOBEC-3A
Name:DNA dC->dU-editing enzyme APOBEC-3A
Synonyms:ABC3A_HUMAN | APOBEC3A | probable DNA dC->dU-editing enzyme APOBEC-3A
Type:Enzyme Catalytic Domain
Mol. Mass.:23013.77
Organism:Homo sapiens (Human)
Description:gi_21955158
Residue:199
Sequence:
MEASPASGPRHLMDPHIFTSNFNNGIGRHKTYLCYEVERLDNGTSVKMDQHRGFLHNQAK
NLLCGFYGRHAELRFLDLVPSLQLDPAQIYRVTWFISWSPCFSWGCAGEVRAFLQENTHV
RLRIFAARIYDYDPLYKEALQMLRDAGAQVSIMTYDEFKHCWDTFVDHQGCPFQPWDGLD
EHSQALSGRLRAILQNQGN
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  Blast E-value cutoff:
BDBM59578
n/a
NameBDBM59578
Synonyms:5-Cyclohexyl-2,4-dihydro-[1,2,4]triazole-3-thione | 5-cyclohexyl-1,2-dihydro-1,2,4-triazole-3-thione | MLS000029617 | SMR000010125 | cid_692347
TypeSmall organic molecule
Emp. Form.C8H13N3S
Mol. Mass.183.274
SMILESS=c1[nH]nc([nH]1)C1CCCCC1
Structure
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