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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Platelet-activating factor receptor | ||
| Ligand | BDBM50002831 | ||
| Substrate/Competitor | n/a | ||
| Ki | 268±n/a nM | ||
| Comments | PDSP_1048 | ||
| Citation |  Tahraoui, L; Floch, A; Cavero, I Functional validation of platelet-activating factor receptor sites characterized biochemically by a specific and reproducible [3H]platelet-activating factor binding in human platelets. J Pharmacol Exp Ther252:1221-7 (1990) [PubMed] | ||
| More Info.: | Get all data from this article | ||
| Platelet-activating factor receptor | |||
| Name: | Platelet-activating factor receptor | ||
| Synonyms: | PAF Platelet activating factor | PAF-R | PAFR | PTAFR | PTAFR_HUMAN | Platelet activating factor receptor | Platelet-activating factor receptor | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 39219.60 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | PAF Platelet activating factor PTAFR HUMAN::P25105 | ||
| Residue: | 342 | ||
| Sequence: |
| ||
| BDBM50002831 | |||
| n/a | |||
| Name | BDBM50002831 | ||
| Synonyms: | (2R,5R)-2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan | (2S,5S)-2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan | (E)-(1R,2R,3R,5R,12S,13R,16S)-16-Hydroxymethyl-5,9,12,13-tetramethyl-4-oxa-tricyclo[10.3.1.0*3,5*]hexadec-8-en-2-ol | (L 652731)2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan | 2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan | 2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan(L-652,731) | 2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan(L-652731) | CHEMBL297624 | L-652731 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C22H28O7 | ||
| Mol. Mass. | 404.4535 | ||
| SMILES | COc1cc(cc(OC)c1OC)[C@@H]1CC[C@H](O1)c1cc(OC)c(OC)c(OC)c1 | ||
| Structure | 
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