| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Histamine H3 receptor |
|---|
| Ligand | BDBM22914 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 2±n/a nM |
|---|
| Comments | PDSP_1847 |
|---|
| Citation |  Arrang, JM; Garbarg, M; Lancelot, JC; Lecomte, JM; Pollard, H; Robba, M; Schunack, W; Schwartz, JC Highly potent and selective ligands for a new class H3 of histamine receptor. Invest Radiol0:0-2 (1988) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Histamine H3 receptor |
|---|
| Name: | Histamine H3 receptor |
|---|
| Synonyms: | HISTAMINE H3 | HRH3 | HRH3_CAVPO | Histamine H3 receptor |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 48753.61 |
|---|
| Organism: | GUINEA PIG |
|---|
| Description: | HISTAMINE H3 HRH3 GUINEA PIG::Q9JI35 |
|---|
| Residue: | 445 |
|---|
| Sequence: | MERAPPDGLMNASGALAGEAAAAAGGARTFSAAWTAVLAALMALLIVATVLGNALVMLAF
VADSSLRTQNNFFLLNLAISDFLVGVFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCT
SSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMVLVWVLAFLLYGPAILSWEYLSG
GSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGARE
AGPDPLPEAQSSPPQPPPGCWGCWPKGQGESMPLHRYGVGEAGPGAEAGEAALGGGSGAA
ASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSL
AIIVSIFGLCWAPYTLLMIIRAACHGHCVPDYWYETSFWLLWANSAVNPVLYPLCHYSFR
RAFTKLLCPQKLKVQPHSSLEHCWK
|
|
|
|---|
| BDBM22914 |
|---|
| n/a |
|---|
| Name | BDBM22914 |
|---|
| Synonyms: | CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide | Thioperamide | US11622967, Compound Thioperamide |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H24N4S |
|---|
| Mol. Mass. | 292.443 |
|---|
| SMILES | S=C(NC1CCCCC1)N1CCC(CC1)c1cnc[nH]1 |
|---|
| Structure | 
|
|---|
Search and Browse
