| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM82042 |
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| Substrate/Competitor | n/a |
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| Ki | 96.8±n/a nM |
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| Comments | PDSP_2501 |
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| Citation |  Bruns, RF; Lu, GH; Pugsley, TA Characterization of the A2 adenosine receptor labeled by [3H]NECA in rat striatal membranes. Mol Pharmacol29:331-46 (1986) [PubMed] |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM82042 |
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| n/a |
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| Name | BDBM82042 |
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| Synonyms: | 1,3-Dimethyl-8-thiophen-2-yl-3,7-dihydro-purine-2,6-dione | 8-(2-Thienyl)theophylline | CAS_267102 | CHEMBL298625 | NSC_267102 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H10N4O2S |
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| Mol. Mass. | 262.288 |
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| SMILES | Cn1c2nc([nH]c2c(=O)n(C)c1=O)-c1cccs1 |
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| Structure | 
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