| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM81971 |
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| Substrate/Competitor | n/a |
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| Ki | 790±n/a nM |
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| Comments | PDSP_755 |
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| Citation |  Leung, E; Kwatra, MM; Hosey, MM; Green, RD Characterization of cardiac A1 adenosine receptors by ligand binding and photoaffinity labeling. J Pharmacol Exp Ther244:1150-6 (1988) [PubMed] |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_CHICK | ADENOSINE A1 | ADORA1 | Adenosine A1 receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36337.19 |
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| Organism: | Chick |
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| Description: | ADENOSINE A1 ADORA1 Chick::P49892 |
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| Residue: | 324 |
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| Sequence: | MAQSVTAFQAAYISIEVLIALVSVPGNILVIWAVKMNQALRDATFCFIVSLAVADVAVGA
LVIPLAIIINIGPQTEFYSCLMMACPVLILTESSILALLAIAVDRYLRVKIPVRYKSVVT
PRRAAVAIACCWIVSFLVGLTPMFGWNNLNKVLGTRDLNVSHSEFVIKCQFETVISMEYM
VYFNFFVWVLPPLLLMLLIYLEVFNLIRTQLNKKVSSSSNDPQKYYGKELKIAKSLALVL
FLFALSWLPLHILNCITLFCPSCKTPHILTYIAIFLTHGNSAMNPIVYAFRIKKFRTAFL
QIWNQYFCCKTNKSSSSSTAETVN
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| BDBM81971 |
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| n/a |
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| Name | BDBM81971 |
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| Synonyms: | 1,3-Diethyl-8-phenyl-3,7-dihydro-purine-2,6-dione | CAS_1328 | CHEMBL11348 | DPX | NSC_1328 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H16N4O2 |
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| Mol. Mass. | 284.3131 |
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| SMILES | CCn1c2nc([nH]c2c(=O)n(CC)c1=O)-c1ccccc1 |
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| Structure | 
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