| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipase A2 |
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| Ligand | BDBM80868 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay |
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| IC50 | 978±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipase A2 |
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| Name: | Phospholipase A2 |
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| Synonyms: | Group IB phospholipase A2 | PA21B_HUMAN | PLA2 | PLA2A | PLA2G1B | PPLA2 | Phosphatidylcholine 2-acylhydrolase 1B | Phospholipase A2 (PLA2) | Phospholipase A2 group 1B | phospholipase A2 precursor |
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| Type: | Protein |
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| Mol. Mass.: | 16364.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P04054 |
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| Residue: | 148 |
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| Sequence: | MKLLVLAVLLTVAAADSGISPRAVWQFRKMIKCVIPGSDPFLEYNNYGCYCGLGGSGTPV
DELDKCCQTHDNCYDQAKKLDSCKFLLDNPYTHTYSYSCSGSAITCSSKNKECEAFICNC
DRNAAICFSKAPYNKAHKNLDTKKYCQS
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| BDBM80868 |
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| n/a |
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| Name | BDBM80868 |
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| Synonyms: | MLS000582413 | N-(3-chloranyl-2-pyrrolidin-1-yl-phenyl)-3-(2-oxidanylidenechromen-3-yl)benzamide | N-(3-chloro-2-pyrrolidin-1-ylphenyl)-3-(2-oxochromen-3-yl)benzamide | N-(3-chloro-2-pyrrolidino-phenyl)-3-(2-ketochromen-3-yl)benzamide | N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-3-(2-oxo-1-benzopyran-3-yl)benzamide | N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-3-(2-oxo-2H-chromen-3-yl)benzamide | SMR000200958 | cid_2301800 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H21ClN2O3 |
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| Mol. Mass. | 444.91 |
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| SMILES | Clc1cccc(NC(=O)c2cccc(c2)-c2cc3ccccc3oc2=O)c1N1CCCC1 |
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| Structure | 
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