| Reaction Details |
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 | Report a problem with these data |
| Target | Aspartyl aminopeptidase |
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| Ligand | BDBM50008434 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_32822 (CHEMBL646473) |
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| Ki | 57000.0±n/a nM |
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| Citation |  Ocain, TD; Rich, DH alpha-Keto amide inhibitors of aminopeptidases. J Med Chem35:451-6 (1992) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Aspartyl aminopeptidase |
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| Name: | Aspartyl aminopeptidase |
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| Synonyms: | ASPEP | Aminopeptidase | Aspartyl aminopeptidase | DAP | DNPEP | DNPEP_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 52436.31 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_32822 |
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| Residue: | 475 |
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| Sequence: | MQVAMNGKARKEAVQTAAKELLKFVNRSPSPFHAVAECRNRLLQAGFSELKETEKWNIKP
ESKYFMTRNSSTIIAFAVGGQYVPGNGFSLIGAHTDSPCLRVKRRSRRSQVGFQQVGVET
YGGGIWSTWFDRDLTLAGRVIVKCPTSGRLEQQLVHVERPILRIPHLAIHLQRNINENFG
PNTEMHLVPILATAIQEELEKGTPEPGPLNAVDERHHSVLMSLLCAHLGLSPKDIVEMEL
CLADTQPAVLGGAYDEFIFAPRLDNLHSCFCALQALIDSCAGPGSLATEPHVRMVTLYDN
EEVGSESAQGAQSLLTELVLRRISASCQHPTAFEEAIPKSFMISADMAHAVHPNYLDKHE
ENHRPLFHKGPVIKVNSKQRYASNAVSEALIREVANKVKVPLQDLMVRNDTPCGTTIGPI
LASRLGLRVLDLGSPQLAMHSIREMACTTGVLQTLTLFKGFFELFPSLSHNLLVD
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| BDBM50008434 |
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| n/a |
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| Name | BDBM50008434 |
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| Synonyms: | 5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acid | CHEMBL140459 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H23NO3 |
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| Mol. Mass. | 277.3587 |
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| SMILES | CC(C)C[C@H](N)C(=O)CC(Cc1ccccc1)C(O)=O |
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| Structure | 
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