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TargetSigma intracellular receptor 2
LigandBDBM50260592
Substrate/Competitorn/a
Meas. Tech.ChEBML_1694032
Ki>1000±n/a nM
Citation Fanter, LMüller, CSchepmann, DBracher, FWünsch, B Chiral-pool synthesis of 1,2,4-trisubstituted 1,4-diazepanes as novel? Bioorg Med Chem25:4778-4799 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma intracellular receptor 2
Name:Sigma intracellular receptor 2
Synonyms:S2r | SGMR2_RAT | Sigma intracellular receptor 2 | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:Protein
Mol. Mass.:20953.88
Organism:Rattus norvegicus (Rat)
Description:Q5U3Y7
Residue:176
Sequence:
MGAVTARRCVEWLLGLYFVSHIPITMFIDLQALLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLFCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAVHTITTLIPILYTILF
EDFSKAIAFKGQRPENFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKFEEKRKKK
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BDBM50260592
n/a
NameBDBM50260592
Synonyms:CHEMBL4081826
TypeSmall organic molecule
Emp. Form.C23H32N2O
Mol. Mass.352.513
SMILESCOc1ccc(CN2CCCN(Cc3ccccc3)[C@H](C2)C(C)C)cc1 |r|
Structure
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