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TargetGlucagon-like peptide 1 receptor
LigandBDBM50266693
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1701195 (CHEMBL4052177)
EC50 0.0440±n/a nM
Citation Evers, AHaack, TLorenz, MBossart, MElvert, RHenkel, BStengelin, SKurz, MGlien, MDudda, ALorenz, KKadereit, DWagner, M Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists. J Med Chem60:4293-4303 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Glucagon-like peptide 1 receptor
Name:Glucagon-like peptide 1 receptor
Synonyms:GLP-1 receptor | GLP-1-R | GLP-1R | GLP1R_MOUSE | Glp1r
Type:PROTEIN
Mol. Mass.:53042.00
Organism:Mus musculus
Description:ChEMBL_598679
Residue:463
Sequence:
MASTPSLLRLALLLLGAVGRAGPRPQGTTVSLSETVQKWREYRRQCQRFLTEAPLLATGL
FCNRTFDDYACWPDGPPGSFVNVSCPWYLPWASSVLQGHVYRFCTAEGLWLHKDNSSLPW
RDLSECEESKRGERNFPEEQLLSLYIIYTVGYALSFSALVIASAILVGFRHLHCTRNYIH
LNLFASFILRALSVFIKDAALKWMYSTAAQQHQWDGLLSYQDSLGCRLVFLLMQYCVAAN
YYWLLVEGVYLYTLLAFSVFSEQRIFKLYLSIGWGVPLLFVIPWGIVKYLYEDEGCWTRN
SNMNYWLIIRLPILFAIGVNFLIFIRVICIVVSKLKANLMCKTDIKCRLAKSTLTLIPLL
GTHEVIFAFVMDEHARGTLRFIKLFTELSFTSFQGLMVAILYCFVNNEVQMEFRKCWERW
RLEHLNIQRDCSMKPLKCPTSSVSSGATVGSSVYAATCQSSYS
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  Blast E-value cutoff:
BDBM50266693
n/a
NameBDBM50266693
Synonyms:CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucagon Emergency Kit | Glucagon Recombinant
TypeSmall organic molecule
Emp. Form.C153H225N43O49S
Mol. Mass.3482.747
SMILESn/a
Structure
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