| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM50269834 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1707354 (CHEMBL4058587) |
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| Ki | >100000±n/a nM |
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| Citation |  Lefin, R; van der Walt, MM; Milne, PJ; Terre'Blanche, G Imidazo[1,2-?]pyridines possess adenosine A Bioorg Med Chem Lett27:3963-3967 (2017) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM50269834 |
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| n/a |
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| Name | BDBM50269834 |
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| Synonyms: | CHEMBL1807290 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H21N3 |
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| Mol. Mass. | 291.3901 |
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| SMILES | C1CCC(CC1)Nc1c(nc2ccccn12)-c1ccccc1 |
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| Structure | 
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