| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM50014265 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_29008 |
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| Ki | 18000±n/a nM |
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| Citation |  Müller, CE; Hide, I; Daly, JW; Rothenhäusler, K; Eger, K 7-Deaza-2-phenyladenines: structure-activity relationships of potent A1 selective adenosine receptor antagonists. J Med Chem33:2822-8 (1990) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM50014265 |
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| n/a |
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| Name | BDBM50014265 |
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| Synonyms: | 5,6-Dimethyl-7-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine | CHEMBL319540 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H14N4 |
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| Mol. Mass. | 238.2878 |
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| SMILES | Cc1c(C)c2c(N)ncnc2n1-c1ccccc1 |
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| Structure | 
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