| Reaction Details |
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 | Report a problem with these data |
| Target | Gastric inhibitory polypeptide receptor |
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| Ligand | BDBM50266693 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1714753 (CHEMBL4124802) |
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| EC50 | >100000±n/a nM |
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| Citation |  Evers, A; Bossart, M; Pfeiffer-Marek, S; Elvert, R; Schreuder, H; Kurz, M; Stengelin, S; Lorenz, M; Herling, A; Konkar, A; Lukasczyk, U; Pfenninger, A; Lorenz, K; Haack, T; Kadereit, D; Wagner, M Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists Specifically Optimized for Multidose Formulations. J Med Chem61:5580-5593 (2018) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Gastric inhibitory polypeptide receptor |
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| Name: | Gastric inhibitory polypeptide receptor |
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| Synonyms: | GIPR | GIPR_HUMAN | Gastric Inhibitory Polypeptide Receptor (GIPR) | Gastric inhibitory polypeptide receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 53173.82 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1518286 |
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| Residue: | 466 |
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| Sequence: | MTTSPILQLLLRLSLCGLLLQRAETGSKGQTAGELYQRWERYRRECQETLAAAEPPSGLA
CNGSFDMYVCWDYAAPNATARASCPWYLPWHHHVAAGFVLRQCGSDGQWGLWRDHTQCEN
PEKNEAFLDQRLILERLQVMYTVGYSLSLATLLLALLILSLFRRLHCTRNYIHINLFTSF
MLRAAAILSRDRLLPRPGPYLGDQALALWNQALAACRTAQIVTQYCVGANYTWLLVEGVY
LHSLLVLVGGSEEGHFRYYLLLGWGAPALFVIPWVIVRYLYENTQCWERNEVKAIWWIIR
TPILMTILINFLIFIRILGILLSKLRTRQMRCRDYRLRLARSTLTLVPLLGVHEVVFAPV
TEEQARGALRFAKLGFEIFLSSFQGFLVSVLYCFINKEVQSEIRRGWHHCRLRRSLGEEQ
RQLPERAFRALPSGSGPGEVPTSRGLSSGTLPGPGNEASRELESYC
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| BDBM50266693 |
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| n/a |
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| Name | BDBM50266693 |
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| Synonyms: | CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucagon Emergency Kit | Glucagon Recombinant |
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| Type | Small organic molecule |
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| Emp. Form. | C153H225N43O49S |
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| Mol. Mass. | 3482.747 |
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| SMILES | n/a |
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| Structure | 
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