Reaction Details |
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Target | Cytosol aminopeptidase [33-68,L62W] |
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Ligand | BDBM50457466 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1759783 (CHEMBL4194791) |
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IC50 | 100±n/a nM |
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Citation | Amin, SA; Adhikari, N; Jha, T Design of Aminopeptidase N Inhibitors as Anti-cancer Agents. J Med Chem61:6468-6490 (2018) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Cytosol aminopeptidase [33-68,L62W] |
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Name: | Cytosol aminopeptidase [33-68,L62W] |
Synonyms: | AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP) |
Type: | Enzyme |
Mol. Mass.: | 4015.44 |
Organism: | Sus scrofa (Pig) |
Description: | P28839[33-68,L62W] |
Residue: | 36 |
Sequence: | TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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BDBM50457466 |
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n/a |
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Name | BDBM50457466 |
Synonyms: | CHEMBL4206158 |
Type | Small organic molecule |
Emp. Form. | C21H30N2O6 |
Mol. Mass. | 406.4727 |
SMILES | CC(C)C[C@@H]([C@H](O)C(=O)NO)C(=O)N[C@H](C(=O)OC1CCCC1)c1ccccc1 |r| |
Structure |
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