| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50458142 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1762409 (CHEMBL4197656) |
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| Ki | 6.1±n/a nM |
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| Citation |  Turnaturi, R; Marrazzo, A; Parenti, C; Pasquinucci, L Benzomorphan scaffold for opioid analgesics and pharmacological tools development: A comprehensive review. Eur J Med Chem148:410-422 (2018) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50458142 |
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| n/a |
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| Name | BDBM50458142 |
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| Synonyms: | CHEMBL4208635 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H26N2O2 |
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| Mol. Mass. | 326.4326 |
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| SMILES | CCC12CCN(CC3CC3)C(C1C)C(=O)c1ccc(NC=O)cc21 |TLB:14:13:11:3.4.5,6:5:11:15.23.13,THB:22:23:11:3.4.5| |
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| Structure | 
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