| Reaction Details |
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 | Report a problem with these data |
| Target | Kappa-type opioid receptor |
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| Ligand | BDBM50458148 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1762416 (CHEMBL4197663) |
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| Ki | 1.3±n/a nM |
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| Citation |  Turnaturi, R; Marrazzo, A; Parenti, C; Pasquinucci, L Benzomorphan scaffold for opioid analgesics and pharmacological tools development: A comprehensive review. Eur J Med Chem148:410-422 (2018) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Kappa-type opioid receptor |
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| Name: | Kappa-type opioid receptor |
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| Synonyms: | Kappa-type opioid receptor | OPRK1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 13196.24 |
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| Organism: | Macaca mulatta |
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| Description: | ChEMBL_117796 |
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| Residue: | 115 |
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| Sequence: | RYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFP
DDDYSWWDLFMKICVFVFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLR
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|
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| BDBM50458148 |
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| n/a |
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| Name | BDBM50458148 |
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| Synonyms: | CHEMBL4214248 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H25NO |
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| Mol. Mass. | 271.3972 |
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| SMILES | [H][C@]12Cc3ccc(O)cc3[C@@](C)(CCN1CCC=C)[C@H]2C |r,THB:8:9:19:12.13.14,15:14:19:3.9.2| |
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| Structure | 
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