| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma intracellular receptor 2 |
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| Ligand | BDBM50466978 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1794681 (CHEMBL4266798) |
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| Ki | 422±n/a nM |
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| Citation |  Zampieri, D; Romano, M; Menegazzi, R; Mamolo, MG New piperidine-based derivatives as sigma receptor ligands. Synthesis and pharmacological evaluation. Bioorg Med Chem Lett28:3206-3209 (2018) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma intracellular receptor 2 |
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| Name: | Sigma intracellular receptor 2 |
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| Synonyms: | S2r | SGMR2_RAT | Sigma intracellular receptor 2 | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97 |
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| Type: | Protein |
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| Mol. Mass.: | 20953.88 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q5U3Y7 |
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| Residue: | 176 |
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| Sequence: | MGAVTARRCVEWLLGLYFVSHIPITMFIDLQALLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLFCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAVHTITTLIPILYTILF
EDFSKAIAFKGQRPENFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKFEEKRKKK
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| BDBM50466978 |
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| n/a |
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| Name | BDBM50466978 |
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| Synonyms: | CHEMBL4284278 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H26N2O |
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| Mol. Mass. | 274.4011 |
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| SMILES | CCN(CC1CCN(Cc2ccccc2)CC1)C(C)=O |
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| Structure | 
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