Reaction Details |
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Target | Melatonin receptor type 1C |
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Ligand | BDBM9019 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_104759 (CHEMBL710991) |
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Ki | 0.176000±n/a nM |
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Citation | Langlois, M; Brémont, B; Shen, S; Poncet, A; Andrieux, J; Sicsic, S; Serraz, I; Mathé-Allainmat, M; Renard, P; Delagrange, P Design and synthesis of new naphthalenic derivatives as ligands for 2-[125I]iodomelatonin binding sites. J Med Chem38:2050-60 (1995) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Melatonin receptor type 1C |
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Name: | Melatonin receptor type 1C |
Synonyms: | CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C |
Type: | PROTEIN |
Mol. Mass.: | 38595.98 |
Organism: | Gallus gallus |
Description: | ChEMBL_104739 |
Residue: | 346 |
Sequence: | MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGN
IFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAI
NRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTV
STSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVV
FVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFR
KEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
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BDBM9019 |
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n/a |
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Name | BDBM9019 |
Synonyms: | CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide |
Type | Small organic molecule |
Emp. Form. | C13H16N2O2 |
Mol. Mass. | 232.2783 |
SMILES | COc1ccc2[nH]cc(CCNC(C)=O)c2c1 |
Structure |
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