| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Melatonin receptor type 1C |
|---|
| Ligand | BDBM50470711 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_104754 (CHEMBL712437) |
|---|
| Ki | 0.055800±n/a nM |
|---|
| Citation |  Garratt, PJ; Jones, R; Tocher, DA; Sugden, D Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines. J Med Chem38:1132-9 (1995) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Melatonin receptor type 1C |
|---|
| Name: | Melatonin receptor type 1C |
|---|
| Synonyms: | CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 38595.98 |
|---|
| Organism: | Gallus gallus |
|---|
| Description: | ChEMBL_104739 |
|---|
| Residue: | 346 |
|---|
| Sequence: | MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGN
IFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAI
NRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTV
STSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVV
FVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFR
KEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
|
|
|
|---|
| BDBM50470711 |
|---|
| n/a |
|---|
| Name | BDBM50470711 |
|---|
| Synonyms: | CHEMBL14403 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H24N2O2 |
|---|
| Mol. Mass. | 336.4275 |
|---|
| SMILES | CCCC(=O)NCCc1c([nH]c2ccc(OC)cc12)-c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
