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TargetSimilar to alpha-tubulin isoform 1
LigandBDBM50472222
Substrate/Competitorn/a
Meas. Tech.ChEMBL_211324 (CHEMBL818983)
IC50 3600±n/a nM
Citation Poncet, JBusquet, MRoux, FPierré, AAtassi, GJouin, P Synthesis and biological activity of chimeric structures derived from the cytotoxic natural compounds dolastatin 10 and dolastatin 15. J Med Chem41:1524-30 (1998) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Similar to alpha-tubulin isoform 1
Name:Similar to alpha-tubulin isoform 1
Synonyms:Similar to alpha-tubulin isoform 1
Type:PROTEIN
Mol. Mass.:10383.05
Organism:Bos taurus
Description:ChEMBL_104716
Residue:99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGK
HVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50472222
n/a
NameBDBM50472222
Synonyms:CHEMBL608244
TypeSmall organic molecule
Emp. Form.C44H69N5O9
Mol. Mass.812.0468
SMILESCC[C@H](C)[C@@H]([C@@H](CC(=O)N1CCC[C@H]1C(=O)O[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc2)C(OC)=CC1=O)OC)N(C)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)C)C(C)C |r,c:36|
Structure
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