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TargetCannabinoid receptor 2
LigandBDBM50072757
Substrate/Competitorn/a
Meas. Tech.ChEMBL_46995 (CHEMBL658964)
Ki 320±n/a nM
Citation Fichera, MCruciani, GBianchi, AMusumarra, G A 3D-QSAR study on the structural requirements for binding to CB(1) and CB(2) cannabinoid receptors. J Med Chem43:2300-9 (2000) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:39690.94
Organism:Homo sapiens (Human)
Description:P34972
Residue:360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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  Blast E-value cutoff:
BDBM50072757
n/a
NameBDBM50072757
Synonyms:(5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-fluoro-ethyl)-amide | CHEMBL74909 | Icosa-5,8,11,14-tetraenoic acid (2-fluoro-ethyl)-amide (0585)
TypeSmall organic molecule
Emp. Form.C22H36FNO
Mol. Mass.349.5257
SMILESCCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)NCCF
Structure
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