| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50072760 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_327124 (CHEMBL864630) |
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| EC50 | 7943±n/a nM |
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| Citation |  Salo, OM; Savinainen, JR; Parkkari, T; Nevalainen, T; Lahtela-Kakkonen, M; Gynther, J; Laitinen, JT; Järvinen, T; Poso, A 3D-QSAR studies on cannabinoid CB1 receptor agonists: G-protein activation as biological data. J Med Chem49:554-66 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52856.55 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | P20272 |
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| Residue: | 473 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAI
AVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHV
FHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCL
MWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILW
KAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPL
LAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTA
QPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50072760 |
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| n/a |
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| Name | BDBM50072760 |
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| Synonyms: | 3-Hydroxy-N-((5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenyl)-propionamide | 3-hydroxy-N-icosa-5,8,11,14-tetraenyl)propanamide | CHEMBL150849 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H39NO2 |
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| Mol. Mass. | 361.5613 |
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| SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCCNC(=O)CCO |
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| Structure | 
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