| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Alpha-2B adrenergic receptor |
|---|
| Ligand | BDBM50118705 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_911054 (CHEMBL3057215) |
|---|
| Ki | 977±n/a nM |
|---|
| Citation |  TBA Med Chem Res13:134-148 (2004) Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Alpha-2B adrenergic receptor |
|---|
| Name: | Alpha-2B adrenergic receptor |
|---|
| Synonyms: | ADA2B_RAT | Adra2b | Adrenergic receptor alpha | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Alpha-2B adrenoceptor | Alpha-2B adrenoreceptor | adrenergic Alpha2B |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 50379.83 |
|---|
| Organism: | NEONATAL RAT |
|---|
| Description: | adrenergic Alpha2B ADRA2B NEONATAL RAT::P19328 |
|---|
| Residue: | 453 |
|---|
| Sequence: | MSGPTMDHQEPYSVQATAAIASAITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLA
AADILVATLIIPFSLANELLGYWYFWRAWCEVYLALDVLFCTSSIVHLCAISLDRYWAVS
RALEYNSKRTPRRIKCIILTVWLIAAVISLPPLIYKGDQRPEPRGLPQCELNQEAWYILA
SSIGSFFAPCLIMILVYLRIYVIAKRSHCRGLGAKRGSGEGESKKPQPVAGGVPTSAKVP
TLVSPLSSVGEANGHPKPPREKEEGETPEDPEARALPPTWSALPRSGQGQKKGTSGATAE
EGDEEDEEEVEECEPQTLPASPASVCNPPLQQPQTSRVLATLRGQVLLGKNVGVASGQWW
RRRTQLSREKRFTFVLAVVIGVFVVCWFPFFFSYSLGAICPQHCKVPHGLFQFFFWIGYC
NSSLNPVIYTVFNQDFRRAFRRILCRPWTQTGW
|
|
|
|---|
| BDBM50118705 |
|---|
| n/a |
|---|
| Name | BDBM50118705 |
|---|
| Synonyms: | ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1H-imidazol-4-ylmethyl)-phenyl]-amide | N-(3-((1H-imidazol-4-yl)methyl)phenyl)ethanesulfonamide | N-[3-(1H-imidazol-4-ylmethyl)-phenyl]ethanesulfonamide |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H15N3O2S |
|---|
| Mol. Mass. | 265.331 |
|---|
| SMILES | CCS(=O)(=O)Nc1cccc(Cc2cnc[nH]2)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
