| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-1B adrenergic receptor |
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| Ligand | BDBM50118705 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_911066 (CHEMBL3056713) |
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| Ki | 891±n/a nM |
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| Citation |  TBA Med Chem Res13:134-148 (2004) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Alpha-1B adrenergic receptor |
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| Name: | Alpha-1B adrenergic receptor |
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| Synonyms: | ADA1B_MESAU | ADRA1B | adrenergic Alpha1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 56514.13 |
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| Organism: | HAMSTER |
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| Description: | adrenergic Alpha1 0 HAMSTER::P18841 |
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| Residue: | 515 |
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| Sequence: | MNPDLDTGHNTSAPAQWGELKDANFTGPNQTSSNSTLPQLDVTRAISVGLVLGAFILFAI
VGNILVILSVACNRHLRTPTNYFIVNLAIADLLLSFTVLPFSATLEVLGYWVLGRIFCDI
WAAVDVLCCTASILSLCAISIDRYIGVRYSLQYPTLVTRRKAILALLSVWVLSTVISIGP
LLGWKEPAPNDDKECGVTEEPFYALFSSLGSFYIPLAVILVMYCRVYIVAKRTTKNLEAG
VMKEMSNSKELTLRIHSKNFHEDTLSSTKAKGHNPRSSIAVKLFKFSREKKAAKTLGIVV
GMFILCWLPFFIALPLGSLFSTLKPPDAVFKVVFWLGYFNSCLNPIIYPCSSKEFKRAFM
RILGCQCRSGRRRRRRRRLGACAYTYRPWTRGGSLERSQSRKDSLDDSGSCMSGSQRTLP
SASPSPGYLGRGAQPPLELCAYPEWKSGALLSLPEPPGRRGRLDSGPLFTFKLLGEPESP
GTEGDASNGGCDATTDLANGQPGFKSNMPLAPGHF
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| BDBM50118705 |
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| n/a |
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| Name | BDBM50118705 |
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| Synonyms: | ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1H-imidazol-4-ylmethyl)-phenyl]-amide | N-(3-((1H-imidazol-4-yl)methyl)phenyl)ethanesulfonamide | N-[3-(1H-imidazol-4-ylmethyl)-phenyl]ethanesulfonamide |
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| Type | Small organic molecule |
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| Emp. Form. | C12H15N3O2S |
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| Mol. Mass. | 265.331 |
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| SMILES | CCS(=O)(=O)Nc1cccc(Cc2cnc[nH]2)c1 |
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| Structure | 
|
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