| Reaction Details |
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 | Report a problem with these data |
| Target | Nicotinic acetylcholine receptor alpha 5 subunit |
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| Ligand | BDBM82070 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_916315 (CHEMBL3081642) |
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| IC50 | 11900±n/a nM |
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| Citation |  Kagabu, S; Kiriyama, K; Nishiwaki, H; Kumamoto, Y; Tada, T; Nishimura, K Asymmetric chloronicotinyl insecticide, 1-[1-(6-chloro-3-pyridyl)ethyl]-2-nitroiminoimidazolidine: preparation, resolution and biological activities toward insects and their nerve preparations. Biosci Biotechnol Biochem67:980-8 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Nicotinic acetylcholine receptor alpha 5 subunit |
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| Name: | Nicotinic acetylcholine receptor alpha 5 subunit |
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| Synonyms: | Nicotinic acetylcholine receptor alpha 5 subunit | nAChRalpha5 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 88489.00 |
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| Organism: | Musca domestica |
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| Description: | ChEMBL_106552 |
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| Residue: | 781 |
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| Sequence: | MMWEMLILWAVHLSLTAIATLYANVRTALSQTAQQIVRAVIAATTLPIIQRIQQQQHETE
KQQQQLQHGKHVEDIHLPAAGARYASASSSRLPPSSADATIWPRAPPELPQTEKLSSAPP
PPSSSSTLLMQTKPAHKKPVHGRNFPPQQKNRMQPVSHLQYQQQQQQQLSLPSPAEPQPQ
HYKQQQQQQGQERLGQQVNINNITSSSNGGNTCSSNSFTATTSIAATTTTSILTLWQHCH
RRYRPHQLLPLLTTKGLNKYSWIFLLIYLNLSAKVCLAGYNEKRLLHDLLDTYNTLERPV
LNESDPLQLSFGLTLMQIIDVDEKNQLLVTNVWLKLEWNDMNLRWNTSDYGGIKDLRIPP
HRIWKPDVLMYNSADEGFDGTYQTNVVVRNNGSCLYVPPGIFKSTCKIDITWFPFDDQRC
EMKFGSWTYDGFQLDLQLQDETGGDISSYVLNGEWELLGVPGKRNEIYYNCCPEPYIDIT
FAIIIRRRTLYYFFNLIIPCVLIASMALLGFTLPPDSGEKLSLGVTILLSLTVFLNMVAE
TMPATSDAVPLLGTYFNCIMFMVASSVVSTILILNYHHRNADTHEMSEWIRVVFLCWLPW
ILRMHRPGRPIIMDFTSTPCSDTSSERKHQILSDVELKERSSKSLLANVLDIDDDFRNVR
PMTPGGTLPHNPAFYRTVYGYLENLQGDDGSIGPIGSTRMPDAVTHHTCIKTQTEYELSL
ILKEIRFITDQLRKEDEENGIANDWKFAAMVVDRLCLIIFTMFAILATIAVLLSAPHVIV
S
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| BDBM82070 |
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| n/a |
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| Name | BDBM82070 |
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| Synonyms: | CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D salicylate | US10667515, Compound (S)-nicotine | US9303017, Nicotine |
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| Type | n/a |
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| Emp. Form. | C10H14N2 |
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| Mol. Mass. | 162.2316 |
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| SMILES | CN1CCC[C@H]1c1cccnc1 |r| |
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| Structure | 
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