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TargetNicotinic acetylcholine receptor alpha 5 subunit
LigandBDBM50488029
Substrate/Competitorn/a
Meas. Tech.ChEMBL_916315 (CHEMBL3081642)
IC50 190±n/a nM
Citation Kagabu, SKiriyama, KNishiwaki, HKumamoto, YTada, TNishimura, K Asymmetric chloronicotinyl insecticide, 1-[1-(6-chloro-3-pyridyl)ethyl]-2-nitroiminoimidazolidine: preparation, resolution and biological activities toward insects and their nerve preparations. Biosci Biotechnol Biochem67:980-8 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Nicotinic acetylcholine receptor alpha 5 subunit
Name:Nicotinic acetylcholine receptor alpha 5 subunit
Synonyms:Nicotinic acetylcholine receptor alpha 5 subunit | nAChRalpha5
Type:PROTEIN
Mol. Mass.:88489.00
Organism:Musca domestica
Description:ChEMBL_106552
Residue:781
Sequence:
MMWEMLILWAVHLSLTAIATLYANVRTALSQTAQQIVRAVIAATTLPIIQRIQQQQHETE
KQQQQLQHGKHVEDIHLPAAGARYASASSSRLPPSSADATIWPRAPPELPQTEKLSSAPP
PPSSSSTLLMQTKPAHKKPVHGRNFPPQQKNRMQPVSHLQYQQQQQQQLSLPSPAEPQPQ
HYKQQQQQQGQERLGQQVNINNITSSSNGGNTCSSNSFTATTSIAATTTTSILTLWQHCH
RRYRPHQLLPLLTTKGLNKYSWIFLLIYLNLSAKVCLAGYNEKRLLHDLLDTYNTLERPV
LNESDPLQLSFGLTLMQIIDVDEKNQLLVTNVWLKLEWNDMNLRWNTSDYGGIKDLRIPP
HRIWKPDVLMYNSADEGFDGTYQTNVVVRNNGSCLYVPPGIFKSTCKIDITWFPFDDQRC
EMKFGSWTYDGFQLDLQLQDETGGDISSYVLNGEWELLGVPGKRNEIYYNCCPEPYIDIT
FAIIIRRRTLYYFFNLIIPCVLIASMALLGFTLPPDSGEKLSLGVTILLSLTVFLNMVAE
TMPATSDAVPLLGTYFNCIMFMVASSVVSTILILNYHHRNADTHEMSEWIRVVFLCWLPW
ILRMHRPGRPIIMDFTSTPCSDTSSERKHQILSDVELKERSSKSLLANVLDIDDDFRNVR
PMTPGGTLPHNPAFYRTVYGYLENLQGDDGSIGPIGSTRMPDAVTHHTCIKTQTEYELSL
ILKEIRFITDQLRKEDEENGIANDWKFAAMVVDRLCLIIFTMFAILATIAVLLSAPHVIV
S
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  Blast E-value cutoff:
BDBM50488029
n/a
NameBDBM50488029
Synonyms:(S)-METHYL-IMIDACLOPRID
TypeSmall organic molecule
Emp. Form.C10H12ClN5O2
Mol. Mass.269.688
SMILESC[C@H](N1CCN\C1=N/[N+]([O-])=O)c1ccc(Cl)nc1 |r|
Structure
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