| Reaction Details |
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 | Report a problem with these data |
| Target | Peroxisome proliferator-activated receptor alpha |
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| Ligand | BDBM50269532 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_933251 (CHEMBL3069175) |
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| IC50 | 270±n/a nM |
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| Citation |  TBA Med Chem Res22:3126-3133 (2013) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Peroxisome proliferator-activated receptor alpha |
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| Name: | Peroxisome proliferator-activated receptor alpha |
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| Synonyms: | NR1C1 | Nuclear receptor subfamily 1 group C member 1 | PPAR | PPAR alpha/gamma | PPAR-alpha | PPARA | PPARA_HUMAN | Peroxisome Proliferator-Activated Receptor alpha | Peroxisome proliferator-activated receptor | Peroxisome proliferator-activated receptor alpha (PPAR alpha) |
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| Type: | Enzyme |
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| Mol. Mass.: | 52222.08 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q07869 |
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| Residue: | 468 |
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| Sequence: | MVDTESPLCPLSPLEAGDLESPLSEEFLQEMGNIQEISQSIGEDSSGSFGFTEYQYLGSC
PGSDGSVITDTLSPASSPSSVTYPVVPGSVDESPSGALNIECRICGDKASGYHYGVHACE
GCKGFFRRTIRLKLVYDKCDRSCKIQKKNRNKCQYCRFHKCLSVGMSHNAIRFGRMPRSE
KAKLKAEILTCEHDIEDSETADLKSLAKRIYEAYLKNFNMNKVKARVILSGKASNNPPFV
IHDMETLCMAEKTLVAKLVANGIQNKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANL
DLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFD
FAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDI
FLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDMY
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| BDBM50269532 |
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| n/a |
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| Name | BDBM50269532 |
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| Synonyms: | (6,9,12)-linolenic acid | (6Z,9Z,12Z)-octadeca-6,9,12-trienoic acid | (Z,Z,Z)-6,9,12-octadecatrienoic acid | CHEMBL464982 | US9061023, gamma-Linolenic acid | all-cis-6,9,12-octadecatrienoic acid | cis-Delta(6,9,12)-octadecatrienoic acid | gamma-linolenic acid | gamolenic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C18H30O2 |
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| Mol. Mass. | 278.4296 |
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| SMILES | CCCCC\C=C/C\C=C/C\C=C/CCCCC(O)=O |
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| Structure | 
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