| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50049394 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_32014 (CHEMBL649050) |
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| Ki | 1720±n/a nM |
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| Citation |  Ji, XD; Melman, N; Jacobson, KA Interactions of flavonoids and other phytochemicals with adenosine receptors. J Med Chem39:781-8 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM50049394 |
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| n/a |
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| Name | BDBM50049394 |
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| Synonyms: | 5,4'-Dihydroxy-6,7-dimethoxyflavone | 5-Hydroxy-2-(4-hydroxy-phenyl)-6,7-dimethoxy-chromen-4-one | 5-hydroxy-2-(4-hydroxyphenyl)-6,7-dimethoxy-4H-chromen-4-one | CHEMBL348436 | Cirsimaritin | cid_188323 | cirsimartin |
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| Type | Small organic molecule |
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| Emp. Form. | C17H14O6 |
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| Mol. Mass. | 314.2895 |
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| SMILES | COc1cc2oc(cc(=O)c2c(O)c1OC)-c1ccc(O)cc1 |
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| Structure | 
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