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TargetCyclin-dependent kinase 1
LigandBDBM50056181
Substrate/Competitorn/a
Meas. Tech.ChEMBL_48699 (CHEMBL657992)
IC50>1000000±n/a nM
Citation Havlícek, LHanus, JVeselý, JLeclerc, SMeijer, LShaw, GStrnad, M Cytokinin-derived cyclin-dependent kinase inhibitors: synthesis and cdc2 inhibitory activity of olomoucine and related compounds. J Med Chem40:408-12 (1997) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cyclin-dependent kinase 1
Name:Cyclin-dependent kinase 1
Synonyms:CDC2 | CDC28A | CDK1 | CDK1_HUMAN | CDKN1 | Cell division control protein 2 homolog | Cell division protein kinase 1 | Cyclin-dependent kinase 1 (CDK1) | P34CDC2 | p34 protein kinase
Type:Enzyme Subunit
Mol. Mass.:34101.08
Organism:Homo sapiens (Human)
Description:P06493
Residue:297
Sequence:
MEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRH
PNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCH
SRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPIRVYTHEVVTLWYRSPEVLLGSAR
YSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNT
FPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFNDLDNQIKKM
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  Blast E-value cutoff:
BDBM50056181
n/a
NameBDBM50056181
Synonyms:Benzyl-(1-methyl-6,9-dihydro-1H-purin-6-yl)-amine | CHEMBL133290
TypeSmall organic molecule
Emp. Form.C13H15N5
Mol. Mass.241.2917
SMILESCN1C=Nc2nc[nH]c2C1NCc1ccccc1 |c:2|
Structure
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