| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A2b |
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| Ligand | BDBM50511941 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1846295 (CHEMBL4346836) |
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| Ki | 8.3±n/a nM |
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| Citation |  Jiang, J; Seel, CJ; Temirak, A; Namasivayam, V; Arridu, A; Schabikowski, J; Baqi, Y; Hinz, S; Hockemeyer, J; Müller, CE A J Med Chem62:4032-4055 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A2b |
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| Name: | Adenosine receptor A2b |
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| Synonyms: | AA2BR_MOUSE | Adenosine A2b receptor | Adora2b |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36130.09 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_11831 |
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| Residue: | 332 |
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| Sequence: | MQLETQDALYVALELVIAALAVAGNVLVCAAVGASSALQTPTNYFLVSLATADVAVGLFA
IPFAITISLGFCTDFHGCLFLACFVLVLTQSSIFSLLAVAVDRYLAIRVPLRYKGLVTGT
RARGIIAVLWVLAFGIGLTPFLGWNSKDSATSNCTELGDGIANKSCCPVTCLFENVVPMS
YMVYFNFFGCVLPPLLIMLVIYIKIFMVACKQLQRMELMDHSRTTLQREIHAAKSLAMIV
GIFALCWLPVHAINCITLFHPALAKDKPKWVMNVAILLSHANSVVNPIVYAYRNRDFRYS
FHKIISRYVLCQAETKGGSGQAGAQSTLSLGL
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| BDBM50511941 |
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| n/a |
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| Name | BDBM50511941 |
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| Synonyms: | CHEMBL4537196 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H27ClN6O4S |
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| Mol. Mass. | 543.038 |
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| SMILES | CCCn1c(=O)n(C)c2nc([nH]c2c1=O)-c1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(Cl)cc1 |
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| Structure | 
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