| Reaction Details |
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 | Report a problem with these data |
| Target | Group 10 secretory phospholipase A2 |
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| Ligand | BDBM50534281 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1928085 (CHEMBL4431157) |
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| IC50 | 2200±n/a nM |
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| Citation |  Giordanetto, F; Pettersen, D; Starke, I; Nordberg, P; Dahlström, M; Knerr, L; Selmi, N; Rosengren, B; Larsson, LO; Sandmark, J; Castaldo, M; Dekker, N; Karlsson, U; Hurt-Camejo, E Discovery of AZD2716: A Novel Secreted Phospholipase A ACS Med Chem Lett7:884-889 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Group 10 secretory phospholipase A2 |
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| Name: | Group 10 secretory phospholipase A2 |
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| Synonyms: | Group X secretory phospholipase A2 | PA2GX_HUMAN | PLA2G10 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 18153.11 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1442449 |
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| Residue: | 165 |
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| Sequence: | MGPLPVCLPIMLLLLLPSLLLLLLLPGPGSGEASRILRVHRRGILELAGTVGCVGPRTPI
AYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGP
AENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD
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| BDBM50534281 |
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| n/a |
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| Name | BDBM50534281 |
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| Synonyms: | CHEMBL4536076 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H13NO |
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| Mol. Mass. | 211.2591 |
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| SMILES | NC(=O)c1ccc(Cc2ccccc2)cc1 |
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| Structure | 
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