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Reaction Details
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TargetSigma intracellular receptor 2
LigandBDBM50562179
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2077638 (CHEMBL4733429)
Ki 3.0±n/a nM
Citation Xie, XYLi, YYMa, WHChen, AFSun, YTLee, JYRiad, AXu, DHMach, RHHuang, YS Synthesis, binding, and functional properties of tetrahydroisoquinolino-2-alkyl phenones as selective ? Eur J Med Chem209:0 (2021) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma intracellular receptor 2
Name:Sigma intracellular receptor 2
Synonyms:S2r | SGMR2_RAT | Sigma intracellular receptor 2 | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:Protein
Mol. Mass.:20953.88
Organism:Rattus norvegicus (Rat)
Description:Q5U3Y7
Residue:176
Sequence:
MGAVTARRCVEWLLGLYFVSHIPITMFIDLQALLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLFCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAVHTITTLIPILYTILF
EDFSKAIAFKGQRPENFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKFEEKRKKK
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BDBM50562179
n/a
NameBDBM50562179
Synonyms:CHEMBL4739972
TypeSmall organic molecule
Emp. Form.C27H37NO7
Mol. Mass.487.5852
SMILESCOc1cc2CCN(CCCCC(=O)c3c(C)c(OC)c(OC)c(OC)c3OC)Cc2cc1OC
Structure
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