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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Delta-type opioid receptor | ||
| Ligand | BDBM50144286 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEBML_147341 | ||
| Ki | 16±n/a nM | ||
| Citation |  Carson, JR; Coats, SJ; Codd, EE; Dax, SL; Lee, J; Martinez, RP; McKown, LA; Anne Neilson, L; Pitis, PM; Wu, WN; Zhang, SP N-alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]benzamides, micro and delta opioid agonists: a micro address. Bioorg Med Chem Lett14:2113-6 (2004) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Delta-type opioid receptor | |||
| Name: | Delta-type opioid receptor | ||
| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 | ||
| Type: | G Protein-Coupled Receptor (GPCR) | ||
| Mol. Mass.: | 40382.98 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. | ||
| Residue: | 372 | ||
| Sequence: |
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| BDBM50144286 | |||
| n/a | |||
| Name | BDBM50144286 | ||
| Synonyms: | CHEMBL306463 | N-Ethyl-4-{[8-(5-methyl-1H-imidazol-4-ylmethyl)-8-aza-bicyclo[3.2.1]oct-3-ylidene]-phenyl-methyl}-benzamide | ||
| Type | Small organic molecule | ||
| Emp. Form. | C28H32N4O | ||
| Mol. Mass. | 440.5799 | ||
| SMILES | CCNC(=O)c1ccc(cc1)C(=C1CC2CCC(C1)N2Cc1[nH]cnc1C)c1ccccc1 |(19.23,1.17,;17.89,1.92,;17.87,3.47,;16.54,4.23,;16.52,5.77,;15.2,3.45,;15.22,1.9,;13.88,1.12,;12.55,1.9,;12.53,3.42,;13.85,4.21,;11.21,1.12,;11.23,-.41,;12.56,-1.19,;12.58,-2.9,;11.87,-1.63,;10.67,-1.63,;9.89,-2.75,;9.89,-1.19,;11.23,-3.51,;11.23,-5.06,;12.56,-5.83,;13.97,-5.22,;15,-6.36,;14.21,-7.68,;12.71,-7.35,;11.58,-8.38,;9.88,1.88,;9.88,3.42,;8.54,4.18,;7.2,3.4,;7.22,1.85,;8.56,1.11,)| | ||
| Structure | 
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