| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide FF receptor 1 |
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| Ligand | BDBM50029188 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2158113 (CHEMBL5042863) |
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| Ki | 0.010000±n/a nM |
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| Citation |  Quillet, R; Schneider, S; Utard, V; Drieu la Rochelle, A; Elhabazi, K; Henningsen, JB; Gizzi, P; Schmitt, M; Kugler, V; Simonneaux, V; Ilien, B; Simonin, F; Bihel, F Identification of an J Med Chem64:7555-7564 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide FF receptor 1 |
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| Name: | Neuropeptide FF receptor 1 |
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| Synonyms: | G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47840.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1474637 |
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| Residue: | 430 |
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| Sequence: | MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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| BDBM50029188 |
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| n/a |
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| Name | BDBM50029188 |
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| Synonyms: | CHEMBL2165920 |
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| Type | Small organic molecule |
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| Emp. Form. | C45H72N14O10 |
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| Mol. Mass. | 969.141 |
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| SMILES | CC(C)C[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)C(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r| |
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| Structure | 
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