| Reaction Details |
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 | Report a problem with these data |
| Target | Baculoviral IAP repeat-containing protein 7 |
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| Ligand | BDBM50588301 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2186645 (CHEMBL5098727) |
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| IC50 | 278±n/a nM |
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| Citation |  Udompholkul, P; Baggio, C; Gambini, L; Alboreggia, G; Pellecchia, M Lysine Covalent Antagonists of Melanoma Inhibitors of Apoptosis Protein. J Med Chem64:16147-16158 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Baculoviral IAP repeat-containing protein 7 |
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| Name: | Baculoviral IAP repeat-containing protein 7 |
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| Synonyms: | BIR3 | BIRC7 | BIRC7_HUMAN | Baculoviral IAP repeat-containing protein 7 | KIAP | LIVIN | MLIAP | RNF50 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 32792.04 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_624591 |
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| Residue: | 298 |
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| Sequence: | MGPKDSAKCLHRGPQPSHWAAGDGPTQERCGPRSLGSPVLGLDTCRAWDHVDGQILGQLR
PLTEEEEEEGAGATLSRGPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQD
KVRCFFCYGGLQSWKRGDDPWTEHAKWFPSCQFLLRSKGRDFVHSVQETHSQLLGSWDPW
EEPEDAAPVAPSVPASGYPELPTPRREVQSESAQEPGGVSPAEAQRAWWVLEPPGARDVE
AQLRRLQEERTCKVCLDRAVSIVFVPCGHLVCAECAPGLQLCPICRAPVRSRVRTFLS
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| BDBM50588301 |
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| n/a |
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| Name | BDBM50588301 |
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| Synonyms: | CHEMBL5195146 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H37N5O8S |
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| Mol. Mass. | 615.698 |
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| SMILES | CN[C@@H](C)C(=O)N[C@@H](CNC(=O)c1cc(ccc1OC)S(O)(=O)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H]1CCc2ccccc12 |r| |
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| Structure | 
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