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TargetType-2 angiotensin II receptor
LigandBDBM50156173
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2211253 (CHEMBL5124202)
Ki 0.400000±n/a nM
Citation Gopalan, GPalo-Nieto, CPetersen, NNHallberg, MLarhed, M Angiotensin II AT2 receptor ligands with phenylthiazole scaffolds. Bioorg Med Chem65:0 (2022) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Type-2 angiotensin II receptor
Name:Type-2 angiotensin II receptor
Synonyms:Angiotensin type II receptor
Type:PROTEIN
Mol. Mass.:15474.49
Organism:Sus scrofa
Description:ChEMBL_1285617
Residue:137
Sequence:
MAFPPEKYAQWSAGIALMKNILGFIIPLVFIATCYFGIRKHLLKTNSYGKNRITRDQVLN
MAAAVVLAFIICWLPFHVLTFLDALAWMGIINSCEVIAVIDLALPFAILLGFTNSCINPF
LYCFVGNRFQQKLRSVF
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  Blast E-value cutoff:
BDBM50156173
n/a
NameBDBM50156173
Synonyms:(1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazol-5-yl)methanol | CHEMBL189568 | butyl (5-isobutylthien-2-yl)sulfonylcarbamate derivative | butyl 3-(4-((1H-imidazol-1-yl)methyl)phenyl)-5-isobutylthiophen-2-ylsulfonylcarbamate
TypeSmall organic molecule
Emp. Form.C23H29N3O4S2
Mol. Mass.475.624
SMILESCCCCOC(=O)NS(=O)(=O)c1sc(CC(C)C)cc1-c1ccc(Cn2ccnc2)cc1
Structure
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